dc.contributor.author |
Baydoun E. |
dc.contributor.author |
Karam M. |
dc.contributor.author |
Atia-Tul-Wahab |
dc.contributor.author |
Khan M.S.A. |
dc.contributor.author |
Ahmad M.S. |
dc.contributor.author |
Samreen |
dc.contributor.author |
Smith C. |
dc.contributor.author |
Abdel-Massih R. |
dc.contributor.author |
Choudhary M.I. |
dc.contributor.editor |
|
dc.date |
2014 |
dc.date.accessioned |
2017-10-03T15:43:32Z |
dc.date.available |
2017-10-03T15:43:32Z |
dc.date.issued |
2014 |
dc.identifier |
10.1016/j.steroids.2014.06.020 |
dc.identifier.isbn |
|
dc.identifier.issn |
|
dc.identifier.uri |
http://hdl.handle.net/10938/12495 |
dc.description.abstract |
Therapeutic potential of nandrolone and its derivatives against leishmaniasis has been studied. A number of derivatives of nandrolone (1) were synthesized through biotransformation. Microbial transformation of nandrolone (1) with Cunninghamella echinulata and Cunninghamella blakesleeana yielded three new metabolites, 10β,12β,17β-trihydroxy-19-nor-4-androsten-3-one (2), 10β,16α,17β-trihydroxy-19-nor-4-androsten-3-one (3), and 6β,10β,17β-trihydroxy-19-nor-4-androsten-3-one (4), along with four known metabolites, 10β,17β-dihydroxy-19-nor-4-androsten-3-one (5), 6β,17β-dihydroxy-19-nor-4-androsten-3-one (6) 10β-hydroxy-19-nor-4-androsten-3,17-dione (7) and 16β,17β- dihydroxy-19-nor-4-androsten-3-one (8). Compounds 1-8 were evaluated for their anti-leishmanial activity. Compounds 1 and 8 showed a significant activity in vitro against Leishmania major. The leishmanicidal potential of compounds 1-8 (IC50 = 32.0 ± 0.5, andgt;100, 77.39 ± 5.52, 70.90 ± 1.16, 54.94 ± 1.01, 80.23 ± 3.39, 61.12 ± 1.39 and 29.55 ± 1.14 μM, respectively) can form the basis for the development of effective therapies against the protozoal tropical disease leishmaniasis. © 2014 Elsevier Inc. All rights reserved. |
dc.format.extent |
|
dc.format.extent |
Pages: (95-100) |
dc.language |
English |
dc.publisher |
Elsevier Inc.; NEW YORK |
dc.relation.ispartof |
Publication Name: Steroids; Publication Year: 2014; Volume: 88; Pages: (95-100); |
dc.relation.ispartofseries |
|
dc.relation.uri |
|
dc.source |
Scopus |
dc.subject.other |
|
dc.title |
Microbial transformation of nandrolone with Cunninghamella echinulata and Cunninghamella blakesleeana and evaluation of leishmaniacidal activity of transformed products |
dc.type |
Article |
dc.contributor.affiliation |
Baydoun, E., Department of Biology, American University of Beirut, Beirut 1107 2020, Lebanon |
dc.contributor.affiliation |
Karam, M., Department of Biology, American University of Beirut, Beirut 1107 2020, Lebanon |
dc.contributor.affiliation |
Atia-Tul-Wahab, Dr. Panjwani Center for Molecular Medicine and Drug Research, International Center for Chemical and Biological Sciences, University of Karachi, Karachi 75270, Pakistan |
dc.contributor.affiliation |
Khan, M.S.A., H.E.J. Research Institute of Chemistry, International Center for Chemical and Biological Sciences, University of Karachi, Karachi 75270, Pakistan |
dc.contributor.affiliation |
Ahmad, M.S., H.E.J. Research Institute of Chemistry, International Center for Chemical and Biological Sciences, University of Karachi, Karachi 75270, Pakistan |
dc.contributor.affiliation |
Samreen, H.E.J. Research Institute of Chemistry, International Center for Chemical and Biological Sciences, University of Karachi, Karachi 75270, Pakistan |
dc.contributor.affiliation |
Smith, C., Department of Biology, American University of Beirut, Beirut 1107 2020, Lebanon |
dc.contributor.affiliation |
Abdel-Massih, R., Department of Biology, University of Balamand, Koura 100, Lebanon |
dc.contributor.affiliation |
Choudhary, M.I., Dr. Panjwani Center for Molecular Medicine and Drug Research, International Center for Chemical and Biological Sciences, University of Karachi, Karachi 75270, Pakistan, H.E.J. Research Institute of Chemistry, International Center for Chemical and Biological Sciences, University of Karachi, Karachi 75270, Pakistan, Department of Biochemistry, Faculty of Science, King Abdulaziz Universisty, Jeddah 21412, Saudi Arabia |
dc.contributor.authorAddress |
Baydoun, E.; Department of Biology, American University of Beirut, Beirut 1107 2020, Lebanon; email: eliasbay@aub.edu.lb |
dc.contributor.authorCorporate |
University: American University of Beirut; Faculty: Faculty of Arts and Sciences; Department: Biology; |
dc.contributor.authorDepartment |
Biology |
dc.contributor.authorDivision |
|
dc.contributor.authorEmail |
eliasbay@aub.edu.lb; iqbal.choudhary@iccs.edu |
dc.contributor.faculty |
Faculty of Arts and Sciences |
dc.contributor.authorInitials |
Baydoun, E |
dc.contributor.authorInitials |
Karam, M |
dc.contributor.authorInitials |
Atia-tul-Wahab |
dc.contributor.authorInitials |
Khan, MSA |
dc.contributor.authorInitials |
Ahmad, MS |
dc.contributor.authorInitials |
Samreen |
dc.contributor.authorInitials |
Smith, C |
dc.contributor.authorInitials |
Abdel-Massih, R |
dc.contributor.authorInitials |
Choudhary, MI |
dc.contributor.authorOrcidID |
|
dc.contributor.authorReprintAddress |
Baydoun, E (reprint author), Amer Univ Beirut, Dept Biol, Beirut 11072020, Lebanon. |
dc.contributor.authorResearcherID |
|
dc.contributor.authorUniversity |
American University of Beirut |
dc.description.cited |
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dc.description.citedCount |
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dc.description.citedTotWOSCount |
0 |
dc.description.citedWOSCount |
0 |
dc.format.extentCount |
6 |
dc.identifier.articleNo |
|
dc.identifier.coden |
STEDA |
dc.identifier.pubmedID |
|
dc.identifier.scopusID |
84905181434 |
dc.identifier.url |
|
dc.publisher.address |
360 PARK AVE SOUTH, NEW YORK, NY 10010-1710 USA |
dc.relation.ispartofConference |
|
dc.relation.ispartofConferenceCode |
|
dc.relation.ispartofConferenceDate |
|
dc.relation.ispartofConferenceHosting |
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dc.relation.ispartofConferenceLoc |
|
dc.relation.ispartofConferenceSponsor |
|
dc.relation.ispartofConferenceTitle |
|
dc.relation.ispartofFundingAgency |
|
dc.relation.ispartOfISOAbbr |
Steroids |
dc.relation.ispartOfIssue |
|
dc.relation.ispartOfPart |
|
dc.relation.ispartofPubTitle |
Steroids |
dc.relation.ispartofPubTitleAbbr |
Steroids |
dc.relation.ispartOfSpecialIssue |
|
dc.relation.ispartOfSuppl |
|
dc.relation.ispartOfVolume |
88 |
dc.source.ID |
WOS:000341549700015 |
dc.type.publication |
Journal |
dc.subject.otherAuthKeyword |
Anabolic compound |
dc.subject.otherAuthKeyword |
Cunninghamella blakesleeana |
dc.subject.otherAuthKeyword |
Cunninghamella echinulata |
dc.subject.otherAuthKeyword |
Leishmania major |
dc.subject.otherAuthKeyword |
Leishmanicidal activity |
dc.subject.otherAuthKeyword |
Nandrolone |
dc.subject.otherChemCAS |
nandrolone, 434-22-0 |
dc.subject.otherIndex |
10beta hydroxy 19 nor 4 androsten 3,17 dione |
dc.subject.otherIndex |
10beta,12beta,17beta trihydroxy 19 nor 4 androsten 3 one |
dc.subject.otherIndex |
10beta,16alpha,17beta trihydroxy 19 nor 4 androsten 3 one |
dc.subject.otherIndex |
10beta,17beta dihydroxy 19 nor 4 androsten 3 one |
dc.subject.otherIndex |
16beta,17beta dihydroxy 19 nor 4 androsten 3 one |
dc.subject.otherIndex |
6beta,10beta,17beta trihydroxy 19 nor 4 androsten 3 one |
dc.subject.otherIndex |
6beta,17beta dihydroxy 19 nor 4 androsten 3 one |
dc.subject.otherIndex |
antileishmanial agent |
dc.subject.otherIndex |
drug metabolite |
dc.subject.otherIndex |
nandrolone |
dc.subject.otherIndex |
unclassified drug |
dc.subject.otherIndex |
antileishmanial activity |
dc.subject.otherIndex |
article |
dc.subject.otherIndex |
biotransformation |
dc.subject.otherIndex |
carbon nuclear magnetic resonance |
dc.subject.otherIndex |
Cunninghamella blakesleeana |
dc.subject.otherIndex |
Cunninghamella echinulata |
dc.subject.otherIndex |
drug activity |
dc.subject.otherIndex |
drug synthesis |
dc.subject.otherIndex |
fermentation |
dc.subject.otherIndex |
in vitro study |
dc.subject.otherIndex |
Leishmania major |
dc.subject.otherIndex |
leishmaniasis |
dc.subject.otherIndex |
nonhuman |
dc.subject.otherIndex |
proton nuclear magnetic resonance |
dc.subject.otherKeywordPlus |
ANABOLIC-STEROIDS |
dc.subject.otherKeywordPlus |
BIOTRANSFORMATION |
dc.subject.otherKeywordPlus |
FUNGI |
dc.subject.otherKeywordPlus |
ELEGANS |
dc.subject.otherWOS |
Biochemistry and Molecular Biology |
dc.subject.otherWOS |
Endocrinology and Metabolism |