dc.contributor.author |
Mills A.D. |
dc.contributor.author |
Nazer M.Z. |
dc.contributor.author |
Haddadin M.J. |
dc.contributor.author |
Kurth M.J. |
dc.contributor.editor |
|
dc.date |
2006 |
dc.date.accessioned |
2017-10-03T15:45:35Z |
dc.date.available |
2017-10-03T15:45:35Z |
dc.date.issued |
2006 |
dc.identifier |
10.1021/jo0524831 |
dc.identifier.isbn |
|
dc.identifier.issn |
00223263 |
dc.identifier.uri |
http://hdl.handle.net/10938/12745 |
dc.description.abstract |
A one-step heterocyclization of o-nitrobenzylamines to 3-alkoxy-2H- indazoles is reported. The electronic nature of the nitrophenyl group, the steric and electronic nature of the R1-functionalized benzylic amine, and the nature of the alcoholic solvent affect the efficiency of this heterocyclization reaction (∼40-90percent). © 2006 American Chemical Society. |
dc.format.extent |
|
dc.format.extent |
Pages: (2687-2689) |
dc.language |
English |
dc.publisher |
WASHINGTON |
dc.relation.ispartof |
Publication Name: Journal of Organic Chemistry; Publication Year: 2006; Volume: 71; no. 7; Pages: (2687-2689); |
dc.relation.ispartofseries |
|
dc.relation.uri |
|
dc.source |
Scopus |
dc.subject.other |
|
dc.title |
N,N-bond-forming heterocyclization: Synthesis of 3-alkoxy-2H-indazoles |
dc.type |
Article |
dc.contributor.affiliation |
Mills, A.D., Department of Chemistry, University of California, One Shields Avenue, Davis, CA 95616, United States |
dc.contributor.affiliation |
Nazer, M.Z., Chemistry Department, Faculty of Science, University of Jordan, Amman, Jordan |
dc.contributor.affiliation |
Haddadin, M.J., Department of Chemistry, American University of Beirut, Beirut, Lebanon |
dc.contributor.affiliation |
Kurth, M.J., Department of Chemistry, University of California, One Shields Avenue, Davis, CA 95616, United States |
dc.contributor.authorAddress |
Kurth, M.J.; Department of Chemistry, University of California, One Shields Avenue, Davis, CA 95616, United States; email: mjkurth@ucdavis.edu |
dc.contributor.authorCorporate |
University: American University of Beirut; Faculty: Faculty of Arts and Sciences; Department: Chemistry; |
dc.contributor.authorDepartment |
Chemistry |
dc.contributor.authorDivision |
|
dc.contributor.authorEmail |
mjkurth@ucdavis.edu |
dc.contributor.faculty |
Faculty of Arts and Sciences |
dc.contributor.authorInitials |
Mills, AD |
dc.contributor.authorInitials |
Nazer, MZ |
dc.contributor.authorInitials |
Haddadin, MJ |
dc.contributor.authorInitials |
Kurth, MJ |
dc.contributor.authorOrcidID |
|
dc.contributor.authorReprintAddress |
Kurth, MJ (reprint author), Univ Calif Davis, Dept Chem, 1 Shields Ave, Davis, CA 95616 USA. |
dc.contributor.authorResearcherID |
|
dc.contributor.authorUniversity |
American University of Beirut |
dc.description.cited |
ARDAKANI M, 1983, J CHEM SOC P1, V10, P2501; Boduszek B, 1997, TETRAHEDRON, V53, P11399, DOI 10.1016-S0040-4020(97)00721-7; BOYER JH, 1986, J CHEM RES SYNOP, V11, P416; Busch V., 1895, J PRAKT CHEM, V2, P404; Butler MS, 2004, J NAT PROD, V67, P2141, DOI 10.1021-np040106y; Campi EM, 1995, AUST J CHEM, V48, P2023, DOI 10.1071-CH9952023; Chen LJ, 1998, TETRAHEDRON LETT, V39, P5351, DOI 10.1016-S0040-4039(98)01068-5; Frontana-Uribe BA, 1999, ACTA CHEM SCAND, V53, P814, DOI 10.3891-acta.chem.scand.53-0814; Frontana-Uribe BA, 1998, TETRAHEDRON, V54, P3197, DOI 10.1016-S0040-4020(98)00058-1; Grimmet M. R., 1997, COMPREHENSIVE ORGANI, V4, P357; HASSNER A, 1994, J HETEROCYCLIC CHEM, V31, P687; JOHNSTON D, 1987, J CHEM SOC P1, V3, P495; KIENZLE F, 1982, EUR J MED CHEM, V17, P547; Kurth MJ, 2005, J ORG CHEM, V70, P1060, DOI 10.1021-jo048153i; Lam PYS, 1998, TETRAHEDRON LETT, V39, P2941, DOI 10.1016-S0040-4039(98)00504-8; MANOUCHEHR AA, 1979, SYNTHESIS-STUTTGART, V4, P308; Paal C., 1891, CHEM BER, V24, P959; Paal C., 1890, CHEM BER, V23, P2640; Padwa A., 1994, PROG HETEROCYCL CHEM, V6, P36; Song JJ, 2000, ORG LETT, V2, P519, DOI 10.1021-ol990409x; Stadlbauer W., 2002, SCI SYNTH, V12, P227; Zhang JF, 2001, TETRAHEDRON LETT, V42, P8405, DOI 10.1016-S0040-4039(01)01842-1 |
dc.description.citedCount |
30 |
dc.description.citedTotWOSCount |
31 |
dc.description.citedWOSCount |
31 |
dc.format.extentCount |
3 |
dc.identifier.articleNo |
|
dc.identifier.coden |
JOCEA |
dc.identifier.pubmedID |
16555821 |
dc.identifier.scopusID |
33645529315 |
dc.identifier.url |
|
dc.publisher.address |
1155 16TH ST, NW, WASHINGTON, DC 20036 USA |
dc.relation.ispartofConference |
|
dc.relation.ispartofConferenceCode |
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dc.relation.ispartofConferenceDate |
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dc.relation.ispartofConferenceHosting |
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dc.relation.ispartofConferenceLoc |
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dc.relation.ispartofConferenceSponsor |
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dc.relation.ispartofConferenceTitle |
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dc.relation.ispartofFundingAgency |
|
dc.relation.ispartOfISOAbbr |
J. Org. Chem. |
dc.relation.ispartOfIssue |
7 |
dc.relation.ispartOfPart |
|
dc.relation.ispartofPubTitle |
Journal of Organic Chemistry |
dc.relation.ispartofPubTitleAbbr |
J. Org. Chem. |
dc.relation.ispartOfSpecialIssue |
|
dc.relation.ispartOfSuppl |
|
dc.relation.ispartOfVolume |
71 |
dc.source.ID |
WOS:000236652200018 |
dc.type.publication |
Journal |
dc.subject.otherAuthKeyword |
|
dc.subject.otherChemCAS |
Indazoles |
dc.subject.otherIndex |
Heterocyclization reaction |
dc.subject.otherIndex |
Indazoles |
dc.subject.otherIndex |
Alcohols |
dc.subject.otherIndex |
Amines |
dc.subject.otherIndex |
Chemical bonds |
dc.subject.otherIndex |
Chemical reactions |
dc.subject.otherIndex |
Organic compounds |
dc.subject.otherIndex |
Solvents |
dc.subject.otherIndex |
Nitrogen compounds |
dc.subject.otherIndex |
aromatic amine |
dc.subject.otherIndex |
benzoic acid derivative |
dc.subject.otherIndex |
indazole derivative |
dc.subject.otherIndex |
o nitrobenzylamine |
dc.subject.otherIndex |
solvent |
dc.subject.otherIndex |
unclassified drug |
dc.subject.otherIndex |
alkylation |
dc.subject.otherIndex |
article |
dc.subject.otherIndex |
arylation |
dc.subject.otherIndex |
chemical bond |
dc.subject.otherIndex |
chemical structure |
dc.subject.otherIndex |
cyclization |
dc.subject.otherIndex |
dielectric constant |
dc.subject.otherIndex |
miscibility |
dc.subject.otherIndex |
reaction analysis |
dc.subject.otherIndex |
solubility |
dc.subject.otherIndex |
synthesis |
dc.subject.otherIndex |
viscosity |
dc.subject.otherIndex |
Cyclization |
dc.subject.otherIndex |
Indazoles |
dc.subject.otherIndex |
Molecular Structure |
dc.subject.otherIndex |
Stereoisomerism |
dc.subject.otherKeywordPlus |
DERIVATIVES |
dc.subject.otherKeywordPlus |
INDAZOLES |
dc.subject.otherWOS |
Chemistry, Organic |